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Prof. Dr. Bedia KAYMAKÇIOĞLU

Yayınlar & Eserler

SCI, SSCI ve AHCI İndekslerine Giren Dergilerde Yayınlanan Makaleler 47

Synthesis and Apoptotic Effects of DNMT Inhibition Targeted Novel Hybrid Molecules Bearing Thiadiazole and Clopidogrel for Cancer Treatment

Polycyclic Aromatic Compounds, 2025 (SCI-Expanded)

Design, synthesis, molecular modeling, in vitro evaluation of novel piperidine-containing hydrazone derivatives as cholinesterase inhibitors

Drug Development Research, Cilt: 85, Sayı: 5, 2024 (SCI-Expanded)

Synthesis, characterization, biological evaluation and in silico studies of novel 1,3,4-thiadiazole derivatives as aromatase inhibitors

Journal of Molecular Structure, Cilt: 1296, 2024 (SCI-Expanded)

Synthesis, Characterization, Molecular Docking Studies and Biological Evaluation of Some Novel 3,5-disubstituted-1-phenyl-4,5-dihydro-1H-pyrazole Derivatives

Current Organic Chemistry, Cilt: 28, Sayı: 3, 2024 (SCI-Expanded)

Synthesis and molecular docking analysis of novel hydrazone and thiosemicarbazide derivatives incorporating a pyrimidine ring: exploring neuroprotective activity

Journal of Biomolecular Structure and Dynamics, 2024 (SCI-Expanded)

Synthesis of Phthalimide Derivatives and Their Insecticidal Activity against Caribbean Fruit Fly, Anastrepha suspensa (Loew)

Biomolecules, Cilt: 13, Sayı: 2, 2023 (SCI-Expanded)

Recent Advances in the Microwave and Ultrasound-assisted Synthesis of Pyrazole Scaffolds

Current Organic Chemistry, Cilt: 27, Sayı: 12, 2023 (SCI-Expanded)

Synthesis, characterization and biological evaluation of some novel sulfonylurea derivatives

Journal of Research in Pharmacy, Cilt: 27, Sayı: 6, 2023 (SCI-Expanded)

Design, synthesis, biological activity evaluation and in silico studies of new nicotinohydrazide derivatives as multi-targeted inhibitors for Alzheimer's disease

Journal of Molecular Structure, Cilt: 1265, 2022 (SCI-Expanded)

N-Substituted Arylidene-3-(Methylsulfonyl)-2-Oxoimidazolidine-1-Carbohydrazide as Cholinesterase Inhibitors: Design, Synthesis, and Molecular Docking Study

Chemistry and Biodiversity, Cilt: 19, Sayı: 8, 2022 (SCI-Expanded)

Induction of Divergent Cell Death Pathways by Urea and Carbohydrazide Derivatives

Anti-Cancer Agents in Medicinal Chemistry, Cilt: 22, Sayı: 9, 2022 (SCI-Expanded)

Synthesis, Biological Evaluation and in Silico Studies of New Pyrazoline Derivatives Bearing Benzo[d]thiazol-2(3H)-one Moiety as Potential Urease Inhibitors

Chemistry and Biodiversity, Cilt: 19, Sayı: 3, 2022 (SCI-Expanded)

Synthesis and anticancer activity of new carbohydrazide derivatives bearing furan moiety

Journal of Research in Pharmacy, Cilt: 26, Sayı: 1, 2022 (SCI-Expanded)

Synthesis of some novel 1,3,4-oxadiazole derivatives and evaluation of their antimicrobial activity

Synthetic Communications, Cilt: 52, Sayı: 6, 2022 (SCI-Expanded)

Synthesis of novel thiosemicarbazone derivatives as antidiabetic agent with enzyme kinetic studies and antioxidant activity

Phosphorus, Sulfur and Silicon and the Related Elements, Cilt: 197, Sayı: 12, 2022 (SCI-Expanded)

Synthesis of novel pyrazoline derivatives and evaluation of their antimicrobial activity

Journal of Research in Pharmacy, Cilt: 26, Sayı: 5, 2022 (SCI-Expanded)

Therapeutic Drug Monitoring in Pediatric Patients Treated with Anti-Tuberculosis Medications by High Performance Liquid Chromatography

Journal of Research in Pharmacy, Cilt: 26, Sayı: 6, 2022 (SCI-Expanded)

Synthesis and Biological Evaluation of Some Hydrazide-Hydrazone Derivatives as Anticancer Agents

Acta Chimica Slovenica, Cilt: 69, Sayı: 4, 2022 (SCI-Expanded)

Synthesis of new hydrazone derivatives and evaluation of their monoamine oxidase inhibitory activity

Bioorganic Chemistry, Cilt: 114, 2021 (SCI-Expanded)

Novel 2,5-disubstituted-1,3,4-oxadiazole derivatives as MAO-B inhibitors: Synthesis, biological evaluation and molecular modeling studies

Bioorganic Chemistry, Cilt: 112, 2021 (SCI-Expanded)

Design, synthesis and biological evaluation of some new 2-Pyrazoline derivatives as potential anticancer agents

Bioorganic Chemistry, Cilt: 102, 2020 (SCI-Expanded)

Synthesis, anticancer evaluation and in silico ADMET studies on urea/thiourea derivatives from gabapentin

Phosphorus, Sulfur and Silicon and the Related Elements, Cilt: 196, Sayı: 4, 2020 (SCI-Expanded)

Design, synthesis and biological screening of novel 1,5-diphenyl-3-(4-(trifluoromethyl)phenyl)-2-pyrazoline derivatives

Acta Chimica Slovenica, Cilt: 67, Sayı: 4, 2020 (SCI-Expanded)

Synthesis and biological evaluation of new pyrazolone Schiff bases as monoamine oxidase and cholinesterase inhibitors

Bioorganic Chemistry, Cilt: 84, 2019 (SCI-Expanded)

Synthesis and anticancer activity of new hydrazide-hydrazones and their Pd(II) complexes

Letters in Drug Design and Discovery, Cilt: 16, Sayı: 5, 2019 (SCI-Expanded)

Design, synthesis, biological evaluation and molecular docking of novel molecules to PARP-1 enzyme

Turkish Journal of Chemistry, Cilt: 43, Sayı: 5, 2019 (SCI-Expanded)

Design, synthesis and evaluation of the biological activities of some new carbohydrazide and urea derivatives Bazı yeni karbohidrazit ve üre türevlerinin tasarımı, sentezi ve biyolojik aktivitelerinin değerlendirilmesi

Turkish Journal of Pharmaceutical Sciences, Cilt: 15, Sayı: 3, 2018 (SCI-Expanded)

Design and evaluation of biological activities of 1,3-oxazolidinone derivatives bearing amide, sulfonamide, and thiourea moieties

Archiv der Pharmazie, Cilt: 351, Sayı: 9, 2018 (SCI-Expanded)

Synthesis, anticancer activity and ADMET studies of N-(5-methyl-1,3,4-thiadiazol-2-yl)-4-[(3-substituted)ureido/thioureido] benzenesulfonamide derivatives

Phosphorus, Sulfur and Silicon and the Related Elements, Cilt: 193, Sayı: 8, 2018 (SCI-Expanded)

Synthesis and structure–activity relationships of carbohydrazides and 1,3,4-oxadiazole derivatives bearing an imidazolidine moiety against the yellow fever and dengue vector, Aedes aegypti

Pest Management Science, Cilt: 74, Sayı: 2, 2018 (SCI-Expanded)

Synthesis and biological evaluation of some new hydrazone derivatives bearing pyrimidine ring as analgesic and anti-inflammatory agents

Acta Poloniae Pharmaceutica - Drug Research, Cilt: 75, Sayı: 5, 2018 (SCI-Expanded)

Synthesis and anticonvulsant activity of some 2-pyrazolines derived from chalcones

Arabian Journal of Chemistry, Cilt: 10, 2017 (SCI-Expanded)

Some N-(5-methyl-1,3,4-thiadiazol-2-yl)-4-[(3-substituted)ureido/thioureido]benzenesulfonamides as carbonic anhydrase I and II inhibitors Karbonik anhidraz I ve II inhibitörü olan bazı N-(5-metil-1,3,4-tiyadiazol-2-il)-4-[(3-sübstitüe)üreido/tiyoüreido] benzensülfonamitler

Marmara Pharmaceutical Journal, Cilt: 21, Sayı: 1, 2017 (SCI-Expanded)

Antiproliferative activity of some tautomeric hydrazones derived from chalcones Şalkonlardan hareketle elde edilen bazı tautomerik hidrazonların antiproliferatif aktiviteleri

Marmara Pharmaceutical Journal, Cilt: 20, Sayı: 2, 2016 (SCI-Expanded)

New piperidine-hydrazone derivatives: Synthesis, biological evaluations and molecular docking studies as AChE and BChE inhibitors

European Journal of Medicinal Chemistry, Cilt: 124, 2016 (SCI-Expanded)

Synthesis and larvicidal and adult topical activity of some hydrazidehydrazone derivatives against Aedes aegypti Bazı hidrazit-hidrazon türevlerinin sentezi ve larvasidal etkileri

Marmara Pharmaceutical Journal, Cilt: 18, Sayı: 3, 2014 (SCI-Expanded)

Biting deterrence and insecticidal activity of hydrazide-hydrazones and their corresponding 3-acetyl-2,5-disubstituted-2,3-dihydro-1,3,4-oxadiazoles against Aedes aegypti

Pest Management Science, Cilt: 69, Sayı: 6, 2013 (SCI-Expanded)

Synthesis and biological activity of substituted urea and thiourea derivatives containing 1,2,4-triazole moieties

Molecules, Cilt: 18, Sayı: 3, 2013 (SCI-Expanded)

Synthesis and biological activity of hydrazide-hydrazones and their corresponding 3-Acetyl-2,5-disubstituted-2,3-dihydro-1,3,4-oxadiazoles

Medicinal Chemistry Research, Cilt: 21, Sayı: 11, 2012 (SCI-Expanded)

Synthesis and evaluation of cytotoxic activities of some substituted isoxazolone derivatives Sübstitüe izoksazolon türevlerinin sentezi ve sitotoksik aktivitelerinin deǧerlendirilmesi

Marmara Pharmaceutical Journal, Cilt: 15, Sayı: 3, 2011 (SCI-Expanded)

Anticonvulsant activity of 3,5-dimethylpyrazole derivatives in animal models

Medicinal Chemistry Research, Cilt: 20, Sayı: 5, 2011 (SCI-Expanded)

Antituberculosis activity of hydrazones derived from 4-fluorobenzoic acid hydrazide

Medicinal Chemistry Research, Cilt: 18, Sayı: 4, 2009 (SCI-Expanded)

Synthesis and anticonvulsant activity of new N-(alkyl/Sub-stituted aryl)-N'-[4-(5-cyclohexylamino)-1,3,4-thiadiazole-2-ylphenyl]thioureas

Archiv der Pharmazie, Cilt: 342, Sayı: 1, 2009 (SCI-Expanded)

Synthesis and antinociceptive-antimicrobial activities of some new amide derivatives of 3,5-di/-and 1,3,5-trimethylpyrazoles

Journal of Enzyme Inhibition and Medicinal Chemistry, Cilt: 23, Sayı: 4, 2008 (SCI-Expanded)

HPLC analysis of in vivo metabolites of 4-nitrobenzoic acid [(5-nitro-2-thiopheneyl)methylene]hydrazide in rats

European Journal of Drug Metabolism and Pharmacokinetics, Cilt: 32, Sayı: 4, 2007 (SCI-Expanded)

High pressure liquid chromatographic analysis of in vivo metabolites of N-(substituted phenyl)-N′-(1,3,5-trimethyl pyrazole-4-yl)thioureas in rats

European Journal of Drug Metabolism and Pharmacokinetics, Cilt: 32, Sayı: 4, 2007 (SCI-Expanded)

Synthesis of some novel azo derivatives of 3,5-dimethly-1-(2-hydroxyethyl) pyrazole as potent analgesic agents

Archiv der Pharmazie, Cilt: 339, Sayı: 5, 2006 (SCI-Expanded)

Hakemli Kongre / Sempozyum Bildiri Kitaplarında Yer Alan Yayınlar 22

Investigation of Novel Sulfonamide-Pyrazoline Hybrid Molecules with Potential Antidiabetic Activity Based on Molecular Modelling Against α-Glucosidase, Aldose Reductase and Dipeptidyl Peptidase 4 (DPP-4),

13. International Drug Chemistry Conference, Türkiye - Antalya, 06 Şubat 2025

Design and Synthesis of New Thoureas Bearing Sulfonamide Moeity as Multi-Targeted Agents for The Treatment of Alzhemer's Disease

13. International Drug Chemistry Conference, Türkiye - Antalya, 06 Şubat 2025

Kanserle tedavisinde yeni bir yaklaşım olan PARP-1 inhibitörlerinin tasarımı ve sentezi

2.Ulusal Marmara Eczacılık Kongresi, Türkiye - İstanbul, 14 - 16 Kasım 2018

Design of potent PARP-1 inhibitors through molecular modeling techniques

54th International Conference on Medicinal Chemistry-RICT 2018, Fransa - Strazburg, 04 - 06 Temmuz 2018

Synthesis and biological evaluation of new schiffbases from antipyrine derivatives

54th International Conference on Medicinal Chemistry-RICT 2018, Fransa - Strazburg, 04 - 06 Temmuz 2018

Discovery of novel urea and carbohydrazide derivatives as potent PARP-1 inhibitors

54th International Conference on Medicinal Chemistry-RICT 2018, Fransa - Strazburg, 04 - 06 Temmuz 2018

Synthesis of novel schiff base derivatives and evaluation oftheir monoamine oxidase inhibitory activity

12th International Symposium on Pharmaceutical Sciences-ISOPS 2018, Türkiye - Ankara, 26 - 29 Haziran 2018

Synthesis, characterization and anti-biofilm activity studies on novel urea/thiourea derivatives

12th International Symposium on Pharmaceutical Sciences-ISOPS 2018, Türkiye - Ankara, 26 - 29 Haziran 2018

Synthesis of novel antipyrine derivatives as cholinesterase inhibitors

12th International Symposium on Pharmaceutical Sciences-ISOPS 2018, Türkiye - Ankara, 26 - 29 Haziran 2018

Design, synthesis and biological evaluation of nicotinate derivatives for cancer therapy

12th International Symposium on Pharmaceutical Sciences-ISOPS 2018, Türkiye - Ankara, 26 - 29 Haziran 2018

Design of Potent Multi-target CAs inhibitors through Pharmacophore Modeling

5th International BAU Drug Design Congress, Türkiye - İstanbul, 19 - 21 Ekim 2017

Pharmacophore Modeling For Design of Multi-Target CAs Inhibitors

UEMK Conferences, Türkiye - Gaziantep, 12 - 13 Ekim 2017

CYTOTOXICITY OF SOME NEW CARBOHYDRAZIDE AND UREADERIVATIVES BEARING PYRIDINE RING

2th International Gazi Pharma Symposium Series, Türkiye - Ankara, 11 - 13 Ekim 2017

SYNTHESIS AND STRUCTURE-ACTIVITY RELATIONSHIPS OFCARBOHYDRAZIDES AND 1,3,4-OXADIAZOLE DERIVATIVESBEARING IMIDAZOLIDINE MOIETY AGAINST THE YELLOWFEVER AND DENGUE VECTOR, AEDES AEGYPTI

2th International Gazi Pharma Symposium Series, Türkiye - Ankara, 11 - 13 Ekim 2017

Synthesis and Anti-inflammatory Activities of Some Pyrimidine Hydrazide Hydrazones

17.Österreichische Chemietega 2017, Joint Meeting of the Swiss and Austrian Chemical Societies, Avusturya - Salzburg, 25 - 28 Eylül 2017

Tüberküloz tedavisi alan çocuk hastalarda yüksek basınçlı sıvı kromatografi yöntemi ile terapötik ilaç izlemi

17.Kromatografi Kongresi (Kromatografi 2017), Türkiye - Çorum, 20 - 22 Eylül 2017

Synthesis, characterization and antimicrobial activity evaluation of new some amide derivatives from isonipecotic acid

IVEK 3RD International Convention of Pharmaceuticals And Pharmacies, Türkiye - İstanbul, 26 - 29 Nisan 2017

Synthesis and Anti-inflammatory Activities of Some Hydrazide Hydrazones of Methyl 4-Chloro-2-Methylthio-5-Pyrimidinecarboxylate

3RD International Convention of Pharmaceuticals And Pharmacies,, Türkiye - İstanbul, 26 - 29 Nisan 2017

Mosquito activity of a series of chalcones and 2 pyrazoline derivatives against Aedes aegypti

The 103rd Annual Meeting of the New Jersey Mosquito Control Association March 2 - 4, 2016 , Golden Nugget – Atlantic City, NJ, Amerika Birleşik Devletleri - New Jersey, 02 - 04 Mart 2016

Synthesis and characterization of some new hydrazone derivatives as potential anticancer agents

2nd International Convention of Pharmaceuticals and Pharmacies, Türkiye - İstanbul, 27 - 29 Kasım 2015

Synthesis and evaluation of some sulfonamide derivatives carrying thiourea moiety as potential inhibitors of human carbonic anhydrase isoenzymes hca I and hca II

International Multidisciplinary Symposium on Drug Research& Development., Türkiye - Ankara, 15 - 17 Ekim 2015

Anticancer activity of some amide derivatives bearing hydrazide moiety

6th BBBB Conference on Pharmaceutical Sciences Strategies to Improve the Quality and Performance of Modern Drug Delivery Systems., Slovenya - Bled, 10 - 12 Eylül 2015